Int J Pharm Pharm Sci, Vol 7, Issue 2 Letter to Editor


USE OF TRANEXAMIC ACID IN MEGALIPOSUCTION

ABHIJIT S. NAIR1, SUNJOY VERMA2

Department of Anesthesiology, Citizens Hospitals, Serilingampally, Hyderabad 500019, Telangana, INDIA.
Email: abhi_9568@yahoo.co.in

Received: 02 Nov 2014 Revised and Accepted: 27 Nov 2014


To

The Editor,

Major surgery and trauma trigger similar haemostatic responses. In both situations severe blood loss presents an extreme challenge to the coagulation system. Part of the response to surgery and trauma is stimulation of clot breakdown i.e. fibrinolysis, which might become pathological in some cases [1]. Antifibrinolytic agents reduce blood loss in patients with both normal and exaggerated fibrinolytic responses to surgery. This happens without apparently increasing the risk of postoperative complications [2]. Tranexamic acid is a synthetic derivative of the amino acid lysine that inhibits fibrinolysis by blocking the lysine binding sites on plasminogen [3]. The similarities of tissue injury after trauma and surgery create a novel model for antifibrinolytic therapy with tranexamic acid. The reason of alarming bleeding in liposuction is factors like smoking, diabetes, hypothyroidism, core hypothermia due to infiltration used by the surgeon during surgery, use of drugs like steroids and non steroidal anti-inflammatory drugs by the patient preoperatively. Liposuction involves lots of fluid administration in the form of crystalloid infiltration by surgeon and crystalloid or colloid infusion by anaesthesiologist. There is a loss of volume in the form of lipoaspirate (aspiration of fat done by the surgeon), blood loss & urine output. The anaesthesiologist has to keep a track of all this and ensure that the patient is neither hypovolemic or hypervolemic, both of which can have detrimental consequences in patient outcome and may exacerbate bleeding [4]. Clinical randomization of an Antifibrinolytic in significant haemorrhage or CRASH 2 trial was a large, randomised placebo controlled trial among trauma victims with or at risk of significant haemorrhage [5]. A loading dose of 1 gm over 10 minutes followed by 1 gm over 8 hours was the protocol used for the patients used in this trial. At doses of 10-20 mg/kg administered before surgery, tranexamic acid has been shown to reduce intra operative blood loss and a reduction in blood transfusion rates during hip and knee arthroplasties [6]. The investigators of CRASH 2 trial provided a note of caution in the form of seizures which may occur with higher doses of tranexamic acid which are 2–10 times than those used in CRASH-2. The proposed mechanism of seizures is due to structural similarity of tranexamic acid to γ-aminobutyric acid which is an inhibitory neurotransmitter. This would be a highly unacceptable complication in liposuction or any form of planned surgery. However, caution is needed before extrapolation of the results of CRASH-2 to surgeries like liposuction until they have been studied in a similarly robust manner.The idea of using tranexamic acid in large volume liposuction is encouraging. However, a randomised control trial is necessary to justify its use and dosage determination in these patients.

ACKNOWLEDGEMENT

Nil

CONFLICTS OF INTEREST

Nil

REFERENCES

  1. Lawson JH, Murphy MP. Challenges for providing effective hemostasis in surgery and trauma. Sem Hematol 2004;41:55–64.
  2. Henry DA, Carless PA, Moxey AJ, O'Connell D, McClelland B, Henderson KM, et al. Anti-fibrinolytic use for minimising perioperative allogeneic blood transfusion. Cochrane Database Syst Rev 2007;4:CD001886.
  3. Okamoto S, Hijikata-Okunomiya A, Wanaka K, Okada Y, Okamoto U. Enzyme controlling medicines: introduction. Semin Thromb Hemostasis 1997;23:493–501.
  4. Sood J, Jayaraman L, Sethi N. Liposuction: anaesthesia challenges. Indian J Anaesth 2011;55(3):220-7.
  5. Shakur H, Roberts I, Bautista R, Caballero J, Coats T, Dewan Y, et al. (CRASH-2 trial collaborators). Effects of tranexamic acid on death, vascular occlusive events, and blood transfusion in trauma patients with significant haemorrhage(CRASH-2): a randomized, placebo-controlled trial. Lancet 2010;376(9734):23-32.
  6. Ralley FE, Berta D, Binns V, Howard J, Naudie DD. One intraoperative dose of tranexamic acid for patients having primary hip or knee arthroplasty. Clin Orthop Relat Res 2010;468(7):1905-11.